Herein, we report an in‐situ mild and metal‐free protocol for thiomethylation of heteroarenes in high yields. The thiomethylation of various chloropurines, nucleosides, and chloroheteroarenes has been accomplished offering easy access to agrochemicals and synthetic molecules useful for drug discovery.

中文翻译：

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氯杂芳烃和氯嘌呤的常温无金属硫甲基化

在此，我们报告了一种原位温和且无金属的杂芳烃硫代甲基化方案，收率高。各种氯嘌呤、核苷和氯杂芳烃的硫甲基化已经完成，为获得可用于药物发现的农用化学品和合成分子提供了方便。